TheDose

Histidine

Also known as L-Histidine, Histidine, (S)-2-Amino-3-(1H-imidazol-4-yl)propanoic acid

CIRPubMed

Safe

CIR Expert Panel says: safe as used in cosmetics.”

Histidine (CAS 71-00-1) is an essential proteinogenic α-amino acid with an imidazole side chain, used in cosmetics as an NMF (natural moisturizing factor) component and humectant. The CIR Expert Panel assessed all 21 α-amino acids used in cosmetics (Burnett et al., IJT 32(Suppl. 4):41S-64S, 2013; PMID 24335967) and explicitly named Histidine in the conclusion as safe in the present practices of use and concentration. The QRT records Histidine with Finding=S (Safe), no qualifying conditions, same citation. Histidine HCl (the hydrochloride salt form) carries the same S finding in the same assessment.


Proteinogenic α-amino acid: essential amino acid (humans cannot synthesize it endogenously) with a basic imidazole side chain conferring metal-chelating and pH-buffering properties

Natural moisturizing factor (NMF) component: free histidine is found in the stratum corneum where it contributes to skin hydration and barrier integrity

Humectant: attracts and binds water via the imidazole nitrogen atoms; the imidazole ring also acts as an antioxidant via metal ion chelation

CIR Expert Panel concluded Histidine is safe as used in cosmetics in the present practices of use and concentration:41-64, 2013; QRT Finding=S)

Used in skin- and hair-conditioning formulations; supports barrier repair in combination with ceramides and fatty acids


Concerns
  • · Histidine is the precursor to histamine via enzymatic decarboxylation; this pathway is biologically significant but not a concern in topical cosmetic application at typical use concentrations
  • · No known sensitization or irritation reported in the CIR group assessment at cosmetic-use concentrations

CIR Expert Panel
Approved
[1]
CIR Expert Panel · Oct 1, 2024Live

CIR Quick Reference Table (October 2024) — Histidine row: Finding=S, Citation=IJT 32(Suppl. 4):41-64, 2013

Histidine | S | | IJT 32(Suppl. 4):41-64, 2013QRT-Update-100824_0.pdf, p. 124
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[2]
Peer-reviewed (PubMed) · Nov 1, 2013

Safety Assessment of α-Amino Acids as Used in Cosmetics (Burnett et al., Int J Toxicol 32(6 Suppl):41S-64S, 2013)

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Sources
2
PubMed citations
1
Evidence quality
moderate
Last verified
Re-reviewed when a new CIR / SCCS opinion publishes.