TheDose

Madecassic Acid

Also known as Madecassic Acid, Brahmic Acid, Centella asiatica triterpene aglycone, 2alpha,3beta,6beta,23-tetrahydroxyurs-12-en-28-oic acid

PubMed

Insufficient data

“No regulator has issued a verdict on this ingredient.”

Madecassic Acid is a pentacyclic ursane-type triterpenoid aglycone isolated from Centella asiatica and the deglycosylated form of madecassoside. Published studies confirm anti-inflammatory, antioxidant, and wound-healing properties; in vitro work at 0–50 µM showed cytoprotective effects without reported toxicity (PMID 27728894). No standalone CIR safety assessment exists for Madecassic Acid as a cosmetic ingredient: direct inspection of the CIR Quick Reference Table (QRT-122017revised072018.pdf) confirms it is absent from the alphabetical M-section, placing it in the same not-assessed status as its glycoside form madecassoside.


Anti-inflammatory: established wound-healing and anti-inflammatory agent; inhibits inflammatory pathways in multiple cell types

Antioxidant/cytoprotective: significantly reduces oxidative stress and endoplasmic reticulum stress in microvascular endothelial cells

Collagen synthesis: stimulates maturation of scar tissue via type I collagen production; supports skin barrier and wound healing

Anticancer potential: evaluated for cell viability inhibition and apoptosis induction in melanoma models as a chemopreventive triterpenoid


Concerns
  • · Contact dermatitis has been documented with topical madecassol preparations containing related Centella asiatica triterpenes; sensitization potential at higher concentrations warrants evaluation

No CIR cosmetic safety assessment on record for Madecassic Acid as an isolated ingredient; the 2015 CIR Centella asiatica group report (IJT) covers 9 whole-plant extracts and cell cultures, not isolated triterpene aglycones

[1]
Peer-reviewed (PubMed) · Dec 1, 2016

Madecassic Acid protects against hypoxia-induced oxidative stress in retinal microvascular endothelial cells via ROS-mediated endoplasmic…

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[2]
Peer-reviewed (PubMed) · Jan 1, 2025

Chemopreventive and Anticancer Activity of Selected Triterpenoids in Melanoma (Dycha et al., Cancers (Basel), 2025)

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[3]
Peer-reviewed (PubMed) · Mar 1, 2023

Therapeutic properties and pharmacological activities of asiaticoside and madecassoside: A review (Bandopadhyay et al., J Cell Mol Med 27…

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Sources
3
PubMed citations
3
Evidence quality
limited
Last verified
Re-reviewed when a new CIR / SCCS opinion publishes.